Broadspectrum substituted benzisoxazole sulfonamide hiv...

Details Broadspectrum substituted benzisoxazole sulfonamide hiv... Broadspectrum substituted benzisoxazole sulfonamide hiv...

C - Chemistry, Metallurgy

07

D

C07D 261/20 (2006.01) A61K 31/423 (2006.01) A61K 31/427 (2006.01) A61P 31/18 (2006.01) C07D 307/00 (2006.01) C07D 413/12 (2006.01) C07D 417/12 (2006.01) C07D 493/04 (2006.01)

Patent

CA 2485903

The present invention concerns the compounds having the formula N-oxides, salts, stereoisomeric forms, racemic mixtures, prodrugs esters and metabolites thereof. It further relates to their use as broadspectrum HIV protease inhibitors, processes for their preparation as well as pharmaceutical compositions and diagnostic kits comprising them. It also concerns combinations thereof with another anti-retroviral agent, and to their use in assays as reference compounds or as reagents.

La présente invention concerne les composés possédant la formules (I), des N-oxydes, des sels, des formes stéréo-isomères, des mélanges racémiques, des promédicaments, des esters et des métabolites correspondants. Ladite invention a également trait à leur utilisation en tant qu'inhibiteurs de la protéase du VIH à large spectre, à des processus liés à leur préparation, ainsi qu'à des compositions pharmaceutiques et à des kits diagnostiques les renfermant. Cette invention a aussi pour objet des combinaisons correspondantes avec un autre agent anti-rétroviral et leur utilisation dans des dosages en tant que composés de référence ou réactifs.

Affiliated with

Also associated with

Rating

Broadspectrum substituted benzisoxazole sulfonamide hiv... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Broadspectrum substituted benzisoxazole sulfonamide hiv..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Broadspectrum substituted benzisoxazole sulfonamide hiv... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1926717