Buprenorphine analogs

Details Buprenorphine analogs Buprenorphine analogs

C - Chemistry, Metallurgy

07

D

C07D 489/12 (2006.01) A61K 31/485 (2006.01) A61P 25/04 (2006.01)

Patent

CA 2731939

The present invention is directed to Buprenor-phine Analog compounds of the Formula I, Formula II or Formula III shown below, wherein R1, R2, R8, R3, R3a, R3b, X, Z and Y are as defined herein., R1 H3CO (I) OCH3 OCH3 (III) Compounds of the Invention are useful for treating pain and other conditions modulated by activity of opioid and ORL1 receptors.

La présente invention porte sur des composés analogues de buprénorphine représentés par la Formule I, la Formule II ou la Formule III présentées ci-dessous, dans lesquelles R1, R2, R8, R3, R3a, R3b, X, Z et Y sont tels que définis dans la description. R1 H3CO (I) OCH3 OCH3 (III). Les composés de l'invention sont utiles pour le traitement de la douleur et d'autres affections modulées par l'activité de récepteurs opioïdes et ORL1.

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