Carboxamide diazepin derivatives, preparation method, use as...

Details Carboxamide diazepin derivatives, preparation method, use as... Carboxamide diazepin derivatives, preparation method, use as...

C - Chemistry, Metallurgy

07

D

C07D 487/04 (2006.01) A61K 31/551 (2006.01) C07K 5/02 (2006.01) C07K 5/078 (2006.01) A61K 38/00 (2006.01)

Patent

CA 2395275

The invention concerns products of formula (I) wherein: R¿1? represents in particular -C(O) -R5, -SO2 -R5 or -C(O) -NR6R5, R2 and R7 are such that either R7 represents a hydrogen atom and R2 is such that the group (a) represents the radical of a natural or non-natural amino acid, or R2 and R7 form together a cycle with the nitrogen and carbon atom whereto they are bound, R3 represents in particular the radical -CH=N2 or -CH2-L-R4, R4 represents in particular a linear or branched alkyl radical, and their additive salts with mineral or organic acids or with mineral or organic bases of said products of formula (I). The invention also concerns the method for preparing said products and their use as medicines.

Produits de formule (I) dans laquelle: R1 représente notamment -C(O) -R5, -SO2- R5 ou -C(O) -NR6R5; R2 et R7 sont tels que soit R7 représente un atome d'hydrogène et R2 est tel que le groupement représente le reste d'un acide aminé naturel ou non naturel, soit R2 et R7 forment un cycle ensemble avec les atomes d'azote et de carbone auxquels ils sont liés; R3 représente notamment le radical -CH=N2 ou -CH2-L-R4; R4 représente notamment un radical alkyle linéaire ou ramifié, ainsi que les sels d'addition avec les acides minéraux et organiques ou avec les bases minérales et organiques desdits produits de formule (I). Procédé de préparation et application à titre de médicaments de ces produits.

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