C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 417/12 (2006.01) A61K 31/405 (2006.01) A61K 31/425 (2006.01) A61K 31/427 (2006.01) A61K 31/44 (2006.01) A61P 1/00 (2006.01) A61P 1/06 (2006.01) A61P 3/04 (2006.01) A61P 25/00 (2006.01) A61P 43/00 (2006.01) C07D 209/42 (2006.01) C07D 277/46 (2006.01) C07D 417/00 (2006.01) C07D 417/02 (2006.01) C07D 417/04 (2006.01) C07D 417/14 (2006.01) C07D 471/04 (2006.01)
Patent
CA 2304397
The invention concerns thiazole derivatives agonist of cholecytokinin (CCK) of formula (I) in which R1 represents a substituted phenyl group; R2 a group selected among CH2-R7, (CH2)2-R7, S-CH2-R7, CH2-S-R7, (C5-C8)alkyl with R7 representing a group (C5-C7)cycloalkyl and R3 a group (A) or (B) with R8 representing a group (CH2)nR15 or (C) and R15 representing COOH or COO(C1-C4)alkyl. The invention also concerns a method for preparing pharmaceutical compositions containing them and their uses for preparing medicines.
La présente invention concerne des dérivés de thiazole agonistes de la cholécystokinine (CCK) de formule (I) dans laquelle R1 représente un groupement phényle substitué, R2 un groupement choisi parmi CH2- R7, (CH2)2-R7, S-CH2-R7, CH2-S-R7, (C5-C8)alkyle avec R7 représentant un groupement (C5-C7)cycloalkyle et R3 un groupement (A) ou (B) avec R8 représentant un groupe (CH2)n R15 ou (C) et R15 représentant COOH ou COO(C1-C4)alkyle. Elle concerne en outre un procédé de préparation des compositions pharmaceutiques les contenant et leurs utilisations pour la préparation de médicaments.
Bignon Eric
Boigegrain Robert
Brodin Roger
Molimard Jean-Charles
Olliero Dominique
Robic
Sanofi-Synthelabo
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