A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 31/407 (2006.01) A61P 9/10 (2006.01) A61P 9/12 (2006.01)
Patent
CA 2535178
The invention relates to compositions and associated methods and uses that contain lolitrem compounds containing the moiety shown in structure (I) or derivatives thereof for ion channel antagonist applications, particularly BK channel antagonist applications. Preferred compounds include lolitrem B, 31- epilolitrem B, lolitriol and lolitrem E. For lolitrem B, a particularly strong and long acting blocking effect is identified.
L'invention concerne des compositions ainsi que des procédés et des utilisations connexes. Les compositions contiennent des composés de lolitrem qui renferment la fraction de structure (I) ou des dérivés correspondants, pour les besoins d'applications antagonistes vis-à-vis de canal ionique, en particulier de type BK. De préférence, les composés renferment : lolitrem B, 31-epilolitrem B, lolitriol et lolitrem E. S'agissant de lolitrem B, on a identifié un effet bloquant particulièrement long et durable.
Dalziel Julie Eleanor
Dunlop James
Munday-Finch Sarah Christine
Agresearch Limited
Ridout & Maybee Llp
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