Compounds having unique cb1 receptor binding selectivity and...

Details Compounds having unique cb1 receptor binding selectivity and... Compounds having unique cb1 receptor binding selectivity and...

C - Chemistry, Metallurgy

07

D

C07D 471/04 (2006.01) A61K 31/415 (2006.01) A61K 31/4745 (2006.01) C07D 231/14 (2006.01) C07D 471/02 (2006.01)

Patent

CA 2482004

Compounds of Formula III (see formula III) are provided that are amide analogs of SR141716A having unique CB1 receptor selectivity and providing WIN sparing binding characteristics, pharmaceutical compositions containing the compounds and their use in a method of treatment of CB1 receptor related disorders, such as obesity, schizophrenia, memory dysfunction and marijuana abuse.

L'invention concerne des composés qui sont des analogues amides de SR141716A présentant une sélectivité de récepteur unique CB1 et assurent des caractéristiques de liaison économisant les WIN. L'invention traite aussi de compositions pharmaceutiques contenant ces composés et de leur utilisation dans un procédé de traitement des troubles liés au récepteur CB1, comme l'obésité, la schizophrénie, les troubles de la mémoire et l'abus de marijuana.

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