Compounds useful as modulators of melanocortin receptors and...

C - Chemistry – Metallurgy – 07 – D

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C07D 403/14 (2006.01) A61K 31/44 (2006.01) A61K 31/445 (2006.01) A61K 31/451 (2006.01) A61K 31/454 (2006.01) A61K 31/4545 (2006.01) A61K 31/505 (2006.01) C07D 401/12 (2006.01) C07D 401/14 (2006.01) C07D 403/12 (2006.01) C07D 405/14 (2006.01) C07D 409/14 (2006.01) C07D 413/14 (2006.01) C07D 417/14 (2006.01) C07D 471/10 (2006.01) C07D 487/04 (2006.01) C07D 491/10 (2006.01) C07D 495/04 (2006.01) C07K 5/06 (2006.01) C07K 5/078 (2006.01) A61K 38/00 (2006.01)

Patent

CA 2438272

Compounds having the formula (I), and pharmaceutically-acceptable salts, hydrates and prodrugs thereof, in which E is formula (II), X is N or CH, W is - NR16R17, -NR16C(=O)R22, -NR16CO2R22, -OR23, or a heteroaryl or heterocyclo group as defined in the specification, and R1 through R12, R16, R17, R22, R23, x, y, and z are as defined in the specification, are useful as modulators of melanocortin receptors, particularly MC-1R and MC-4R.

L'invention concerne des composés de formule (I) et des sels, des hydrates et des promédicaments acceptables sur le plan pharmaceutique de ceux-ci, dans laquelle E est de formule (II), X désigne N ou CH, W représente -NR¿16?R¿17?, -NR¿16?C(=O)R¿22?, -NR¿16?CO¿2?R¿22?, -OR¿23?, ou un groupe hétéroaryle ou hétérocycle tel que défini dans la description, et R¿1? à R¿12?, R¿16?, R¿17?, R¿22?, R¿23?, x, y, et z sont tels que définis dans la description. De tels composés sont utiles comme modulateurs des récepteurs de la mélanocortine, notamment MC-1R et MC-4R.

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