Cyclipostins, process for their preparation and use thereof

Details Cyclipostins, process for their preparation and use thereof Cyclipostins, process for their preparation and use thereof

C - Chemistry, Metallurgy

12

N

C12N 1/20 (2006.01) A61K 31/665 (2006.01) A61P 3/10 (2006.01) C07F 9/6574 (2006.01) C12P 9/00 (2006.01) C12P 17/18 (2006.01)

Patent

CA 2407808

The invention relates to compounds of the general formula (I), wherein R1, R2, E, X1, X2 and X3 have the definitions in this application, obtained by the cultivation of the Streptomyces species HAG 004107 (DSM 13381) and to the physiologically compatible salts and chemical equivalents of said compounds. The invention also relates to a method for producing the cyclipostins and their physiologically compatible salts and chemical equivalents as medicaments, in particular as inhibitors of lipases, and to pharmaceutical preparations containing cyclipostin or a physiologically compatible salt or equivalent thereof.

L'invention concerne des composés de formule générale (I), dans laquelle R?1¿, R?2¿, E, X¿1?, X¿2? et X¿3? ont la signification mentionnée, pouvant être obtenus par culture d'espèces Streptomyces HAG 004107 (DSM 13381), ainsi que leurs sels et équivalents chimiques compatibles physiologiquement. L'invention concerne également un procédé de production de cyclipostines, le micro-organisme HAB 004107 (DSM 13381), l'utilisation de la cyclipostine et de ses sels et équivalents chimiques compatibles physiologiquement, en tant que médicaments, notamment en tant qu'inhibiteurs de lipases, ainsi que des préparations pharmaceutiques présentant contenant de la cyclipostine ou un sel ou équivalent compatibles physiologiquement de celle-ci.

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