Extended triterpene derivatives

Details Extended triterpene derivatives Extended triterpene derivatives

C - Chemistry, Metallurgy

07

J

C07J 63/00 (2006.01) A61K 31/56 (2006.01) A61K 31/58 (2006.01) A61P 31/12 (2006.01) A61P 31/18 (2006.01) C07J 53/00 (2006.01)

Patent

CA 2668452

The present invention concerns novel pharmaceutically active triterpene derivatives, pharmaceutical compositions containing the same, their use as medicaments, and the use of the compounds for the manufacture of specific medicaments. The present invention also concerns a method of treatment involving administration of the compounds. Specifically, the compounds are derivatives of betulinic acid having substitutions at one or more of the C-3, C2-8 and C-19 positions as further described herein. The novel compounds are useful as antiretroviral agents. In particular, the novel compounds are useful for the treatment of Human Immunodeficiency Virus (HIV).

La présente invention concerne de nouveaux dérivés de triterpène pharmaceutiquement actifs, des compositions pharmaceutiques les contenant, leur utilisation en tant que médicaments et l'utilisation des composés pour la fabrication de médicaments spécifiques. La présente invention concerne également un procédé de traitement comprenant l'administration des composés. Les composés sont spécifiquement des dérivés d'acide bétulinique ayant des substitutions au niveau d'une ou plusieurs des positions C-3, C2-8 et C-19 tel que décrit plus en détails dans le présent document. Les nouveaux composés sont utiles en tant qu'agents antirétroviraux. Les nouveaux composés sont notamment utiles pour le traitement du virus de l'immunodéficience humaine (VIH).

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