Flt3 inhibitors for immune suppression

A - Human Necessities – 61 – K

Patent

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A61K 38/54 (2006.01)

Patent

CA 2574150

New methods are provided for suppressing the immune system and for treating immune related disorders. Therapies of the invention include administration of an FLT3 inhibitor compound to a subject in need thereof, such as a subject suffering from organ rejection, bone marrow transplant rejection, acquired immune deficiency syndrome, arthritis, aplastic anemia, graft-versus-host disease, Graves' disease, established experimental allergic encephalitomyelitis, multiple sclerosis, lupus, or a neurological disorder. Methods are also provided for screening therapeutic agents for treating immune disorders, including the use of a mouse having an elevated level of FLT3 receptor activity.

La présente invention concerne de nouvelles techniques permettant de déprimer le système immunitaire et de traiter des troubles associés à l'immunité. Des thérapies de cette invention consistent à administrer un composé inhibiteur de FLT3 à un sujet nécessitant un traitement, tel qu'un sujet souffrant d'un rejet d'organe, d'un rejet de transplantation de moelle épinière, d'un syndrome de déficience immune acquise, d'arthrite, d'anémie aplasique, d'une maladie hôte dirigée contre le greffon, de la maladie de Graves, d'encéphalitomyélite allergique expérimentale établie, de sclérose en plaques, du lupus ou d'un trouble neurologique. Cette invention concerne aussi des techniques de recherche d'agents thérapeutiques qui permettant de traiter des troubles immunitaires, comprenant l'utilisation d'une souris possédant un niveau élevé d'activité du récepteur FLT3.

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