C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 471/04 (2006.01) A61K 31/437 (2006.01) A61K 31/444 (2006.01) A61K 31/496 (2006.01) A61K 31/506 (2006.01) A61K 31/5377 (2006.01) C07D 519/00 (2006.01)
Patent
CA 2636946
The present invention is directed to certain fused triazole compounds which are useful as neurokinin-1 (NK-I) receptor antagonists, and inhibitors of tachykinin and in particular substance P- The invention is also concerned with pharmaceutical formulations comprising these compounds as active ingredients and the use of the compounds and their formulations in the treatment of certain disorders, including emesis, urinary incontinence, depression, and anxiety.
La présente invention concerne certains composés de triazoles fusionnés qui sont utiles comme antagonistes des récepteurs de la neurokinine 1 (NK-I), ainsi que comme inhibiteurs de la tachykinine et en particulier de la substance P. L'invention concerne également des formulations pharmaceutiques comprenant ces composés en tant que principes actifs, ainsi que l'utilisation des composés et de leurs formulations dans le traitement de certains troubles, comprenant les vomissements, l'incontinence urinaire, la dépression et l'anxiété.
Devita Robert J.
Young Jonathan R.
Merck And Co. Inc.
Norton Rose Canada S.e.n.c.r.l.,s.r.l./llp
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