Kappa opioid receptor ligands

Details Kappa opioid receptor ligands Kappa opioid receptor ligands

C - Chemistry, Metallurgy

07

D

C07D 401/12 (2006.01) A61K 31/4725 (2006.01) A61P 25/04 (2006.01)

Patent

CA 2433603

Kappa opioid receptor antagonists are provided that yield significant improvements in functional binding assays to kappa opioid receptors relative to nor-BNI, and the use of these antagonists in treatment of disease states that are ameliorated by binding of the kappa opioid receptor such as heroin or cocaine addictions. These kappa opioid receptors have the formula: (see formula 1).

L'invention concerne des antagonistes du récepteur de kappa opioïdes permettant d'améliorer considérablement les essais fonctionnels de fixation à des récepteurs de kappa opioïdes concernant nor-BNI, ainsi que l'utilisation de ces antagonistes pour traiter des maladies améliorées par la fixation du récepteur de kappa opioïdes, telles que des dépendances à l'héroïne ou à la cocaïne.

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