Lactam-containing compounds and derivatives thereof as...

Details Lactam-containing compounds and derivatives thereof as... Lactam-containing compounds and derivatives thereof as...

C - Chemistry, Metallurgy

07

D

C07D 471/04 (2006.01) A61K 31/4545 (2006.01) A61P 7/02 (2006.01) A61P 9/10 (2006.01)

Patent

CA 2461202

The present application describes lactam-containing compounds and derivatives thereof of Formula I: P4-P-M-M4 or pharmaceutically acceptable salt forms thereof, wherein ring P, if present is a 5-7 membered carbocycle or heterocycle and ring M is a 5-7 membered carbocycle or heterocycle. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.

La présente invention concerne des composés contenant du lactame et des dérivés correspondants de formule (I) : P¿4?-P-M-M¿4? ou des formes de sels associées acceptables sur le plan pharmaceutique. Dans cette formule, l'anneau P, s'il est présent, représente un hétérocycle ou un carbocycle doté de 5 à 7 éléments et l'anneau M représente un hétérocycle ou un carbocycle doté de 5 à 7 éléments. On utilise les composés de cette invention en tant qu'inhibiteurs des sérines protéases similaires à la trypsine, notamment le facteur Xa.

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