C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 487/04 (2006.01) A61K 31/407 (2006.01) A61P 19/00 (2006.01) A61P 29/00 (2006.01) C07D 273/00 (2006.01) C07H 17/08 (2006.01)
Patent
CA 2615581
The present invention relates to macrolide conjugates of pyrrolizine and indolizine derivatives with macrocyclic antibiotics and derivatives thereof. The macrolide conjugates are potent inhibitors of 5-lipoxygenase and cyclooxygenase and are therefore suitable to treat disorders of the rheumatic type and to prevent allergically induced diseases. The macrolide conjugates have significantly enhanced potency and efficacy.
La présente invention concerne des conjugués macrolides de dérivés de pyrrolizine et d'indolizine avec des antibiotiques macrocycliques et leurs dérivés. Les conjugués macrolides sont de puissants inhibiteurs de la 5-lipoxygénase et de la cyclooxygénase et sont donc appropriés pour traiter des troubles de type rhumatismal et pour empêcher des maladies provoquées par des allergies. Les conjugués macrolides ont une puissance et une efficacité significativement améliorées.
Albrecht Wolfgang
Burnet Michael
Gutke Hans-Juergen
Laufer Stefan
Deeth Williams Wall Llp
Merckle Gmbh
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