Metalloprotease inhibitors containing a heterocyclic moiety

Details Metalloprotease inhibitors containing a heterocyclic moiety Metalloprotease inhibitors containing a heterocyclic moiety

C - Chemistry, Metallurgy

07

D

C07D 413/12 (2006.01) A61K 31/536 (2006.01)

Patent

CA 2680173

The present invention relates generally to pharmaceutical agents containing a heterocyclic moiety, and in particular, to heterocyclic metalloprotease inhibiting compounds. More particularly, the present invention provides a new class of heterocyclic MMP-13 inhibiting compounds with a benzoxazinone moiety, that exhibit an increased potency and selectivity in relation to currently known MMP-13 inhibitors.

De manière générale, l'invention concerne des agents pharmaceutiques contenant une fraction hétérocyclique, et en particulier, des composés inhibiteurs de métalloprotéase hétérocycliques. Plus particulièrement, la présente invention fournit une nouvelle catégorie de composés inhibiteurs de MMP-13 hétérocycliques pourvus d'une fraction de benzoxazinone, qui présentent une efficacité et une sélectivité accrues par rapport aux inhibiteurs de MMP-13 actuellement connus.

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