Method for producing an optically active azolyl-.alpha.,...

C - Chemistry – Metallurgy – 07 – D

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

260/313, 260/602

C07D 249/08 (2006.01) C07C 91/22 (1985.01) C07C 103/30 (1985.01)

Patent

CA 1218661

ABSTRACT OF THE DISCLOSURE: The present invention relates to a method for producing optically active alcohol derivatives, which are useful as fungicides, herbicides or plant growth regulators, represented by the formula, Image wherein R1 represents a C3-C8 cycloalkyl group, a halogen- substituted C3-C8 cycloalkyl group, a C5-C8 cycloalkenyl group or a halogen-substituted C5-C8 cycloalkenyl group, or a phenyl group which may be substituted with at least one member selected from the group consisting of a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a cyano group, a C1-C4 alkoxyl group, a phenoxy group and a phenyl group, R2 represents a 1,2,4- triazol-1-yl group and a mark * means an asymmetric carbon, by carrying out the asymmetric reduction of a ketone compound represented by the formula, Image wherein R1 and R2 have the same meanings as above, with a boron hydride-reducing agent (a boron hydride type compound) modified with an optically active amino alcohol represented by the formula, Image wherein R3 represents a C1-C8 alkyl, C6-C10 aryl or C7-C11 aralkyl group, R4 represents a hydrogen atom or a C1-C6 alkyl or C7-C16 aralkyl group, R5 represents a hydrogen atom, a C1-C10 alkyl or C7-C16 aralkyl group, or a C6-C18 aryl group which may be substituted with at least one of C1-C6 alkyl and C1-C6 alkoxyl group, and a mark * has the same meaning as above, in the presence or absence of an acid; and also relates to the boron hydride type compound and its production method comprising reacting the above optically active amino alcohol with a boron hydride com- pound.

455667

LandOfFree

Say what you really think

Search LandOfFree.com for Canadian inventors and patents. Rate them and share your experience with other people.

Rating

Method for producing an optically active azolyl-.alpha.,... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Method for producing an optically active azolyl-.alpha.,..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Method for producing an optically active azolyl-.alpha.,... will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFCA-PAI-O-1215852

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.