Method for producing n-substituted 3.beta.-aminonortropanes

Details Method for producing n-substituted 3.beta.-aminonortropanes Method for producing n-substituted 3.beta.-aminonortropanes

C - Chemistry, Metallurgy

07

D

C07D 451/04 (2006.01)

Patent

CA 2542110

The invention relates to a method for producing, on the basis of the corresponding 3-oxonortropane or the corresponding 3.alpha.-aminonortropane, N- substituted 3.beta.-aminonortropanes of formula (I), wherein R1 is defined as in the claim. According to the inventive method, the starting compounds are converted to the corresponding imines by means of an arylmethylamine or an arylaldehyde, said imines are tautomerized or isomerized and then hydrolyzed. The invention also relates to the novel compounds of formula (V), wherein R1 and Ar are defined as in the claims.

L'invention concerne un procédé servant à produire des 3.beta.-aminonortropanes N-substitués de formule (I), dans laquelle R?1¿ a la signification indiquée dans les revendications, à partir du 3-oxonortropane correspondant ou du 3.alpha.-aminonortropane correspondant. Selon l'invention, on transforme ces derniers avec une méthylamine arylique ou un aldéhyde arylique en imines correspondants, on tautomérise ou on isomérise ces derniers, puis on les hydrolyse. L'invention concerne également les nouveaux composés de formule (V), dans laquelle R?1¿ et Ar ont les significations indiquées dans les revendications.

Affiliated with

Also associated with

Rating

Method for producing n-substituted 3.beta.-aminonortropanes does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Method for producing n-substituted 3.beta.-aminonortropanes, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Method for producing n-substituted 3.beta.-aminonortropanes will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1918258