Mu-opiate receptor peptides

Details Mu-opiate receptor peptides Mu-opiate receptor peptides

C - Chemistry, Metallurgy

07

K

C07K 5/107 (2006.01) A61K 38/07 (2006.01) A61K 38/00 (2006.01)

Patent

CA 2284547

This invention relates to certain peptides and linear and cyclic analogs thereof that bind to the mu(morphine) opiate receptor with higher affinity, selectivity and potency than currently available peptides. This invention also relates to pharmaceutical preparations containing an effective amount of the peptides or salts thereof, and methods for providing analgesia, relief from gastrointestinal disorders such as diarrhea, and therapy for drug dependence containing a pharmaceutically effective amount of the peptides.

L'invention porte sur certains peptides et leurs analogues linéaires et cycliques se fixant au récepteur du mu-opiate (de morphine) avec une plus grande affinité, sélectivité et puissance que les peptides actuellement disponibles. L'invention porte également sur des préparations pharmaceutiques contenant une quantité efficace de ces peptides ou de leurs sels, et sur des procédés générateurs d'analgésie, de soulagement des troubles gastro-intestinaux tels que la diarrhée, et de thérapie de la pharmacodépendance, consistant à administrer une quantité à efficacité pharmaceutique de ces peptides.

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