C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 417/06 (2006.01) A61K 31/445 (2006.01) A61K 31/4535 (2006.01) A61K 31/454 (2006.01) A61P 3/04 (2006.01) C07D 211/26 (2006.01) C07D 401/06 (2006.01) C07D 401/12 (2006.01) C07D 401/14 (2006.01) C07D 409/06 (2006.01) C07D 417/12 (2006.01)
Patent
CA 2483806
The present invention relates to compounds, which comprise a 4-substituted piperidine ring linked to a substituted or unsubstituted hydrocarbyl ring. The compounds, including all enatiomeric and diasteriomeric forms and pharmaceutically acceptable salts thereof, have the formula: (I): Wherein preferably R is substituted aryl, W1 is a carbocyclic unit, and W2 is a heteroatom comprising unit. The compounds are melanocortin receptor ligands useful in the treatment of eating disorders.
La présente invention concerne des composés comprenant un noyau pipéridine substitué en position 4 et lié à un noyau hydrocarbyle non substitué. Ces composés, y compris leurs formes énantiomères et diastéréoisomères et leurs sels pharmaceutiquement acceptables, sont représentés par la formule (I), dans laquelle, de préférence, R est aryle substitué, W?1¿ est une unité carbocyclique et W?2¿ est une unité comprenant un hétéroatome. Lesdits composés sont des ligands du récepteur de la mélanocortine utiles dans le traitement de troubles de l'alimentation.
Ebetino Frank Hallock
Liu Xuewei
Mumin Rashid Naeem
Solinsky Mark Gregory
Wos John August
The Procter & Gamble Company
Torys Llp
LandOfFree
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