New aminopropylphosphinic acids

Details New aminopropylphosphinic acids New aminopropylphosphinic acids

C - Chemistry, Metallurgy

07

F

C07F 9/30 (2006.01) A61K 31/662 (2006.01) C07F 9/48 (2006.01)

Patent

CA 2397583

Novel compounds of formula (I), with the exception of i) the racemate of (3-amino-2-hydroxypropyl)phosphinic acid; and ii)(2R/S, 3R)-(3-amino-2-hydroxybutyl)phosphinic acid, having affinity to one or more GABA B receptors, their pharmaceutically acceptable salts, solvates and stereoisomers, as well as processes for their preparation, pharmaceutical compositions containing said therapeutically active compounds and the use of said active compounds in therapy.

L'invention porte sur des nouveaux composés de formule (I), à l'exception i) du racémique de l'acide (3-amino-2-hydroxypropyl)phosphinique; et ii) de l'acide (2R/S, 3R)-(3-amino-2-hydroxybutyl)phosphinique, et qui présentent une affinité avec un ou plusieurs récepteurs du GABA¿B?. L'invention porte également sur leurs sels, solvates et stéréoisomères pharmacocompatibles, sur leur procédé de préparation, et sur des préparations pharmaceutiques contenant ces composés à pouvoir thérapeutique et leur utilisation à des fins de thérapie.

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