New carboxylic acid amides,the preparation thereof and their...

Details New carboxylic acid amides,the preparation thereof and their... New carboxylic acid amides,the preparation thereof and their...

C - Chemistry, Metallurgy

07

D

C07D 235/14 (2006.01) A61K 31/4184 (2006.01) A61P 7/02 (2006.01) C07D 209/00 (2006.01) C07D 209/14 (2006.01) C07D 215/12 (2006.01) C07D 221/00 (2006.01) C07D 231/00 (2006.01) C07D 235/00 (2006.01) C07D 235/16 (2006.01) C07D 239/00 (2006.01) C07D 277/00 (2006.01) C07D 333/00 (2006.01) C07D 401/06 (2006.01) C07D 401/12 (2006.01) C07D 401/14 (2006.01) C07D 403/06 (2006.01) C07D 403/12 (2006.01) C07D 403/14 (2006.01) C07D 409/06 (2006.01) C07D 409/14 (2006.01) C07D 413/12 (2006.01) C07D 417/06 (2006.01) C07D 41

Patent

CA 2510846

The invention relates to novel substituted carboxamides of general formula (I), in which A, B and R1 to R5 are as defined in claim 1, the tautomers, enantiomers, diastereomers, mixtures and salts thereof, in particular the physiologically-acceptable salts thereof with inorganic acids or bases which have useful properties. The compounds of the general formula I as above the tautomers, enantiomers, diastereomers, mixtures and salts thereof, in particular the physiologically-acceptable salts thereof with inorganic acids or bases and the stereoisomers thereof which have useful pharmacological properties, in particular an antithrombotic effect and a factor Xa-inhibiting effect.

La présente invention concerne de nouveaux amides d'acide carboxylique substitués de formule générale (I), dans laquelle A, B et R?1¿ à R?5¿ sont tels que définis dans la revendication 1, leurs tautomères, leurs énantiomères, leurs diastéréomères, leurs mélanges et leurs sels, en particulier leurs sels physiologiquement acceptables à acides ou bases inorganiques ou organiques, qui présentent de précieuses caractéristiques. Les composés de la formule générale I susmentionnée ainsi que leurs tautomères, leurs énantiomères, leurs diastéréomères, leurs mélanges et leurs sels, en particulier leurs sels physiologiquement acceptables à acides ou bases inorganiques ou organiques, et leurs stéréoisomères présentent de précieuses caractéristiques pharmacologiques, en particulier un effet antithrombotique et un effet inhibiteur de facteur Xa.

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