New isosteric peptides

Details New isosteric peptides New isosteric peptides

C - Chemistry, Metallurgy

07

K

C07K 5/08 (2006.01) A61K 38/06 (2006.01) C07K 5/065 (2006.01) A61K 38/00 (2006.01)

Patent

CA 2116527

2116527 9305069 PCTABS00020 The invention relates to new competitive inhibitors of thrombin, their synthesis, pharmaceutical compositions containing the compounds as active ingredients, and the use of the compounds as anticoagulants for prophylaxis and treatment of thromboembolic diseases, according to formula (1), wherein A represents -CH2-, -CH=CH-, -CH2-CH2- or -CH2-CH2-CH2-; Y represents O or S(O)p, where p is 0, 1 or 2; R1, R2, R3, R3A, R4 and m are defined as in the claims, either as such or in the form of a physiologically acceptable salt and including stereoisomers.

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