New lh-rh antagonists with improved effectiveness

Details New lh-rh antagonists with improved effectiveness New lh-rh antagonists with improved effectiveness

C - Chemistry, Metallurgy

07

K

C07K 7/23 (2006.01) A61K 31/16 (2006.01) A61K 31/27 (2006.01) A61K 31/275 (2006.01) A61K 31/33 (2006.01) A61K 38/09 (2006.01) C07C 257/18 (2006.01) C07C 271/22 (2006.01) C07D 207/27 (2006.01) C07D 209/08 (2006.01) C07D 211/14 (2006.01) C07D 213/56 (2006.01) C07D 213/60 (2006.01) C07D 213/61 (2006.01) C07D 213/64 (2006.01) C07D 213/75 (2006.01) C07D 213/80 (2006.01) C07D 213/84 (2006.01) C07D 215/22 (2006.01) C07D 231/56 (2006.01) C07D 233/26 (2006.01) C07D 233/32 (2006.01) C07D 233/61 (2006.01) C07D 233/64

Patent

CA 2238570

New LH-RH antagonists are disclosed, in particular peptidomimetics and peptides modified in a side chain, their salts with pharmaceutically acceptable acids and a process for preparing these LH-RH antagonists and their salts. The disclosed peptides represent analogues of the luteinising hormone releasing hormone (LH-RH). The disclosed compounds have a high antagonistic power and are free of undesirable side effects, in particular edematogenic effects.

L'invention concerne de nouveaux antagonistes de l'hormone libérant l'hormone lutéinisante (LH-RH), notamment des agents peptidomimétiques et des peptides modifiés dans une chaîne latérale, les sels de ceux-ci avec des acides pharmaceutiquement acceptables et un procédé de préparation des antagonistes de LH-RH et de leurs sels. Ces peptides constituent des analogues de l'hormone libérant l'hormone lutéinisante (LH-RH). Ces composés sont fortement antagonistes et dépourvus d'effets secondaires indésirables, tout particulièrement d'effets oedématogènes.

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