C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 209/04 (2006.01) A61K 31/404 (2006.01) A61K 31/416 (2006.01) A61P 3/10 (2006.01) C07D 401/04 (2006.01) C07D 401/14 (2006.01) C07D 403/04 (2006.01) C07D 403/14 (2006.01)
Patent
CA 2678382
The present invention relates to substituted arylsulphonylglycines of general formula wherein R, R4, X, Y, Z and m are defined as in claim 1, the tautomers, enantiomers, diastereomers, mixtures thereof and salts thereof, which have valuable pharmacological properties, particularly the suppression of the interaction of glycogen phosphorylase a with the GL subunit of glycogen- associated protein phosphatase 1 (PP1 ), and their use as pharmaceutical compositions.
La présente invention concerne des arylsulphonylglycines substituées de formule générale (I), dans laquelle: R, R4, X, Y, Z et m sont tels que définis dans la revendication 1, leurs tautomères, énantiomères, diastéréoisomères, des mélanges de ceux-ci ainsi que leurs sels, ayant de précieuses propriétés pharmacologiques, notamment la suppression de l'interaction de la glycogène phosphorylase avec la sous-unité GL de la protéine phosphatase 1 associée (PP1), et leur utilisation en tant que compositions pharmaceutiques.
Eckhardt Matthias
Langkopf Elke
Pautsch Alexander
Schoelch Corinna
Schuler-Metz Annette
Boehringer Ingelheim International Gmbh
Fetherstonhaugh & Co.
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