Novel 2,3-benzodiazepine derivatives and pharmaceutical...

Details Novel 2,3-benzodiazepine derivatives and pharmaceutical... Novel 2,3-benzodiazepine derivatives and pharmaceutical...

C - Chemistry, Metallurgy

07

D

C07D 243/02 (2006.01) A61K 31/551 (2006.01) A61P 25/00 (2006.01)

Patent

CA 2431761

The invention refers to novel 2,3-benzodiazepine derivatives of formula (I) and pharmaceutical compositions containing the same as the active ingredient. The novel compounds have antipasmodic, muscle relaxant and neuroprotective activities. In formula I; X represents a hydrogen atom, a chloro atom or a methoxy group; Y stands for a hydrogen atom or a halo atom; Z means a methyl group or a chloro atom; R is a C~1-4 alkyl group or a group of the formula - NR1~R~2, wherein R1~ and R2~ represent, independently, a hydrogen atom, a C~1- 4 alkyl group, a C~1-4 alkoxy group or a C3-6~ cycloalkyl group.

L'invention concerne de nouveaux dérivés de 2,3-benzodiazépine représentés par la formule (I) ainsi que des compositions pharmaceutiques contenant lesdits dérivés comme matière active. Ces nouveaux composés présentent des activités antispasmodiques, myorelaxantes et neuroprotectrices. Dans la formule I; X représente hydrogène, chloro ou un groupe méthoxy; Y représente hydrogène ou halo; Z représente un groupe méthyle ou chloro; R représente un groupe alkyle C1-4 ou un groupe représenté par la formule -NR<1>R2, dans laquelle R<1> et R<2> représentent, indépendamment, hydrogène, un groupe alkyle C1-4, un groupe alcoxy C1-4 ou un groupe cycloalkyle C<3-6>.

Affiliated with

Also associated with

Rating

Novel 2,3-benzodiazepine derivatives and pharmaceutical... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Novel 2,3-benzodiazepine derivatives and pharmaceutical..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Novel 2,3-benzodiazepine derivatives and pharmaceutical... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1379046