Novel 3-c(o)r substituted 10-cyclohexylbenzoyl...

C - Chemistry – Metallurgy – 07 – D

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C07D 487/04 (2006.01) A61K 31/5517 (2006.01) A61P 5/10 (2006.01) A61P 15/06 (2006.01) C07D 521/00 (2006.01)

Patent

CA 2443556

The present invention provides novel tricyclic benzodiazepine carboxamides compounds and methods and pharmaceutical compositions utilizing them for the treatment and/or prevention and/or suppression of disorders which may be remedied or alleviated by oxytocin antagonist activity, including prevention and/or suppression of preterm labor, suppression of labor at term prior to caesarean delivery, and for the treatment of dysmenorrhea. These compounds are also useful in enhancing fertility rates, enhancing survival rates and synchronizing estrus in farm animals; and may be useful in the prevention and treatmraent of disfunctions of the oxytocin system in the central nervous system including obsessive compulsive disorder (OCD) and neuropsychiatric disorders.

L'invention concerne de nouveaux composés de carboxamides benzodiazépines tricycliques, des procédés et des compositions pharmaceutiques les utilisant dans le traitement et/ou la prévention et/ou l'élimination de troubles pouvant être soignés ou soulagés par l'activité de l'antagoniste d'oxytocine, notamment dans la prévention et/ou la réduction d'accouchements prématurés, dans la réduction d'accouchements à terme avant l'accouchement par césarienne, et dans le traitement de la dysménorrhée. Ces composés sont également utiles dans l'augmentation du taux de fécondité, du taux de survie et dans la synchronisation de l'oestrus des animaux d'élevage. Il peuvent aussi être utilisés dans la prévention et le traitement de dysfonctionnements du système de l'oxytocine se trouvant dans le système nerveux central, notamment les troubles obsessionnels-compulsifs (TOC) et les troubles neuropsychiatriques.

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