A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 39/385 (2006.01) A61K 39/00 (2006.01) A61K 47/48 (2006.01)
Patent
CA 2377524
The present invention discloses novel complex molecules useful as anti- allergic agents. These complex molecules include in particular, peptidic or peptidomimetic molecules, having a first segment which is competent for cell penetration and a second segment which is able to reduce or abolish mast cell degranulation, and in particular to reduce or abolish allergy mediators such as histamine secretion from mast cells. Specific examples of peptides with the desired activity are disclosed.
La présente invention concerne de nouvelles molécules complexes utiles en tant que nouveaux agents antiallergiques. Ces molécules complexes comprennent en particulier des molécules peptidiques ou peptidomimétiques comportant un premier segment qui est capable de pénétrer dans les cellules et un deuxième segment qui est capable de réduire ou supprimer la dégranulation des mastocytes, et plus particulièrement de réduire ou de supprimer des médiateurs de l'allergie tels que la sécrétion d'histamine produite par les mastocytes. Des exemples spécifiques de peptides présentant l'activité désirée sont présentés.
Eisenberg Ronit
Raz Tamar
Allergene Ltd.
Ramot At Tel-Aviv University Ltd.
Ridout & Maybee Llp
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