C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 209/34 (2006.01) A61K 31/404 (2006.01)
Patent
CA 2559115
The invention relates to aryl-containing 5-acylindolinones of general formula (I) in which R1 to R3 are defined as in Claims 1 to 7, the tautomers, enantiomers, diastereomers, mixtures and salts thereof, all of which having valuable pharmacological properties, particularly an inhibitory effect upon protein kinases, particularly an inhibitory effect upon the activity of glycogen synthase kinase (GSK-3).
La présente invention concerne des 5-acylindolinones contenant aryle, de formule générale (I) dans laquelle R?1¿ à R?3¿ sont tels que définis dans les revendications 1 à 7, leurs tautomères, leurs énantiomères, leurs diastéréomères, des mélanges desdites substances et leurs sels, qui présentent des propriétés pharmacologiques précieuses, en particulier un effet inhibiteur des protéines kinases, et spécifiquement un effet inhibiteur de l'activité de la glycogène synthase kinase (GSK-3).
Heckel Armin
Hoerer Stefan
Kley Joerg
Roth Gerald Juergen
Uphues Ingo
Boehringer Ingelheim International Gmbh
Fetherstonhaugh & Co.
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