Novel heteropyrrole analogs acting on cannabinoid receptors

Details Novel heteropyrrole analogs acting on cannabinoid receptors Novel heteropyrrole analogs acting on cannabinoid receptors

A - Human Necessities

61

K

A61K 31/41 (2006.01) C07D 249/08 (2006.01)

Patent

CA 2594488

Disclosed are biologically active hetero pyrrole analogs such as imidazoles, thiazoles, oxazoles and pyrazoles capable of interacting with the CB1 and/or the CB2 cannabinoid receptors. One aspect discloses hetero pyrrole analogs acting as antagonists for the CB1 and/or the CB2 receptors. Another aspect discloses hetero pyrrole analogs having selectivity for the CB1 or CB2 cannabinoid receptor. Also disclosed are pharmaceutical preparations employing the disclosed analogs and methods of administering therapeutically effective amounts of the disclosed analogs to provide a physiological effect.

L'invention concerne des analogues d'hétéropyrroles biologiquement actifs tels que des imidazoles, des thiazoles, des oxazoles et des pyrazoles pouvant interagir avec les récepteurs cannabinoïdes CB1 et/ou CB2. Dans un aspect, l'invention concerne des analogues d'hétéropyrroles agissant en tant qu'agonistes des récepteurs CB1 et/ou CB2. Dans un autre aspect, l'invention concerne des analogues d'hétéropyrroles présentant une sélectivité pour le récepteur cannabinoïde CB1 ou CB2. L'invention concerne également des préparations pharmaceutiques faisant appel aux analogues de l'invention ainsi que des méthodes d'administration de quantités thérapeutiquement efficaces des analogues de l'invention afin d'obtenir un effet physiologique.

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