Novel peptide derivatives having thiazolyl-alanine residue

Details Novel peptide derivatives having thiazolyl-alanine residue Novel peptide derivatives having thiazolyl-alanine residue

C - Chemistry, Metallurgy

07

K

C07K 5/097 (2006.01) A61K 38/05 (2006.01) A61K 38/06 (2006.01) C07D 207/28 (2006.01) C07D 277/02 (2006.01) C07D 277/24 (2006.01) C07D 417/06 (2006.01) C07D 417/14 (2006.01) C07K 5/02 (2006.01) C07K 5/078 (2006.01) C07K 5/117 (2006.01) A61K 38/00 (2006.01)

Patent

CA 2264268

The compounds having superior activity to known TRH and its derivatives in view of the activation of the central nervous system, for example, sustained acetylcholine releasing action, anti-reserpine action and locomotor increment activity was provided. A peptide derivative of the formula (I): (See formula I) its pharmaceutically acceptable salt, or hydrate thereof.

L'invention concerne des dérivés de peptides représentés par la formule générale (I), des sels pharmacologiquement acceptables de ces derniers, ou des hydrates de ces derniers. Ces composés présentent des effets d'activation centrale améliorés, tels qu'un effet retard de la libération de l'acétylcholine, un effet antiréserpine et un effet d'augmentation de la motilité spontanée par rapport aux dérivés connus de TRH et à la TRH.

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