Novel therapeutic agents that modulate estrogen receptors

Details Novel therapeutic agents that modulate estrogen receptors Novel therapeutic agents that modulate estrogen receptors

A - Human Necessities

61

K

A61K 31/42 (2006.01) A61K 31/535 (2006.01) A61K 38/00 (2006.01) A61K 38/02 (2006.01) A61K 38/16 (2006.01) A61K 39/00 (2006.01) A61K 39/395 (2006.01) A61K 39/44 (2006.01) A61K 51/00 (2006.01) C07B 61/00 (2006.01) C07C 215/60 (2006.01) C07C 217/08 (2006.01) C07C 323/62 (2006.01) C07D 211/42 (2006.01) C07D 211/56 (2006.01) C07D 213/74 (2006.01) C07D 213/80 (2006.01) C07D 263/32 (2006.01) C07D 263/34 (2006.01) C07D 265/30 (2006.01) C07D 265/32 (2006.01) C07D 271/06 (2006.01) C07D 277/24 (2006.01) C07D 277/28 (2

Patent

CA 2319497

Disclosed are novel multi-binding compounds (agents) which bind estrogen receptors. The compounds of this invention comprise a plurality of ligands each of which can bind to such receptors thereby modulating the biological processes/functions thereof. Each of the ligands is covalently attached to a linker or linkers which may be the same or different to provide for the multi- binding compound. The linker is selected such that the multi-binding compound so constructed demonstrates increased modulation of the biological processes mediated by the estrogen receptors.

L'invention se rapporte à de nouveaux composés (agents) à liaisons multiples, qui se lient aux récepteurs d'oestrogènes. Ces composés comprennent plusieurs ligands susceptibles de se lier chacun à ces récepteurs dans le but de moduler leurs fonctions/processus biologiques. Chacun de ces ligands est lié de manière covalente à une ou plusieurs séquences de liaison pouvant être identiques ou différentes de manière à former le composé à liaisons multiples. Ladite séquence de liaison est sélectionnée de sorte que le composé à liaisons multiples ainsi formé présente une activité accrue de modulation des processus biologiques dont la médiation est assurée par le récepteur d'oestrogènes.

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