C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 513/04 (2006.01) A61K 31/429 (2006.01) A61K 31/435 (2006.01) A61K 31/4439 (2006.01) A61K 31/454 (2006.01) A61K 31/5383 (2006.01) A61P 9/10 (2006.01) A61P 25/28 (2006.01) A61P 43/00 (2006.01)
Patent
CA 2365419
Novel thiazolo[3,2-a]benzimidazole derivatives represented by general formula (I), which act specifically on metabotropic glutamate receptors and are useful as drugs; and novel compounds useful as intermediates for the synthesis of the derivatives wherein, R1 is optionally substituted carbamoyl, carbonyl, oxy, amino, carbonylamino, or the like; R2 is hydrogen, lower alkyl, or the like; and R3, R4 and R5 are each independently hydrogen, lower alkyl, or the like.
L'invention concerne de nouveaux nouveaux dérivés de thiazolo[3,2-a]benzimidazole de formule générale (I) agissant particulièrement sur les récepteurs du glutamate métabotropique et servant de médicament. L'invention concerne aussi de nouveaux composés utiles comme intermédiaires pour la synthèse des dérivés de formule (I) dans laquelle R1 est éventuellement un carbamoyle, carbonyle, oxy, amino, carbonylamino substitué ou analogue ; R2 désigne un hydrogène, alkyle inférieur ou analogue ; et R3, R4, et R5 désignent chacun séparément un hydrogène, alkyle inférieur ou analogue.
Hayashibe Satoshi
Itahana Hirotsune
Kamikubo Takashi
Kohara Atsuyuki
Maeno Kyoichi
Dennison Associates
Yamanouchi Pharmaceutical Co. Ltd.
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