Opiate agonists and antagonists

Details Opiate agonists and antagonists Opiate agonists and antagonists

C - Chemistry, Metallurgy

07

D

260/237.6

C07D 489/08 (2006.01) A61K 31/47 (2006.01) A61K 31/485 (2006.01) C07D 221/28 (2006.01) C07D 489/02 (2006.01) C07D 519/00 (2006.01)

Patent

CA 1258674

ABSTRACT OF THE DISCLOSURE Dihydromorphinone compound of the general formula HDM=N-R wherein HDM is Image where * indicates binding carbon R1 is an optionally substituted alkyl, alkylene, cycloalkyl, or cycloalkylene R2 is OH or H R3 is OH or OCH3 and R is N=R4, N-R4, Image NN=R4 R4 is an optionally substituted alkyl, alkylene, cycloalkyl, cycloalkylene, aryl, heterocycloalkyl, hetero- cycloalkylene, or alkenyl, and n is 1-10. This compound is useful for irreversibly blocking opiate receptor binding.

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