Optically active tetrahydronaphthalene derivative

Details Optically active tetrahydronaphthalene derivative Optically active tetrahydronaphthalene derivative

C - Chemistry, Metallurgy

07

D

C07D 401/12 (2006.01) A61K 31/4439 (2006.01) A61P 1/16 (2006.01) A61P 1/18 (2006.01) A61P 9/10 (2006.01) A61P 11/00 (2006.01) A61P 13/12 (2006.01) A61P 17/06 (2006.01) A61P 19/02 (2006.01) A61P 25/28 (2006.01) A61P 29/00 (2006.01) A61P 31/04 (2006.01) A61P 37/06 (2006.01) A61P 37/08 (2006.01) C07D 231/12 (2006.01) C07D 401/14 (2006.01)

Patent

CA 2596993

Compound that as compared with the racemate thereof, is highly enhanced in not only C5a receptor antagonistic activity but also extent of bioavailability, represented by the formula (I). Further, there are provided its pharmacologically acceptable salts, or hydrates or solvates thereof.

La présente invention concerne un composé qui, par comparaison avec son racémate, présente non seulement une activité antagoniste du récepteur du C5a fortement amplifiée mais également un degré de biodisponibilité fortement accru. Ce composé est représenté par la formule: [Formule Chimique 1] (I). L'invention concerne en outre les sels, les hydrates ou les solvates pharmacologiquement acceptables de ce composé.

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