C - Chemistry – Metallurgy – 07 – K
Patent
C - Chemistry, Metallurgy
07
K
C07K 7/18 (2006.01) A61K 38/10 (2006.01) C07K 5/078 (2006.01) A61K 38/00 (2006.01)
Patent
CA 2273190
The invention concerns a pseudopeptide compounds selected among the set constituted by (i) the compounds of formula (I) in which: A1 represents a single bond, D-Arg or L-Lys; A2 represents L-Pro or trans-4-hydroxy-L-Pro (4Hyp); A3 represents L-Phe or L-thienylalanine (Thi); Y represents a hydrogen atom or a C1-C3 alkyl group; X represents a sulphur or oxygen atom; and (ii) their additive salts. The invention also concerns the preparation and use of this compound and its additive salts in therapy.
La présente invention a trait à un composé pseudopeptide qui est choisi parmi l'ensemble constitué par: (i) les composés de formule (I) dans laquelle A¿1? représente une simple liaison, D-Arg ou L-Lys, A¿2? représente L-Pro ou trans-4-hydroxy-L-Pro (4Hyp), A¿3? représente L-Phe ou L-thiénylalanine (Thi), Y représente un atome d'hydrogène ou un groupe alkyle en C¿1?-C¿3?, X représente un atome de soufre ou d'oxygène; et, (ii) leurs sels d'addition. Elle concerne également la préparation et l'utilisation de ce composé et de ses sels d'addition d'acide en thérapeutique.
Amblard Muriel
Daffix Isabelle
Dodey Pierre
Luccarini Jean-Michel
Martinez Jean
Fournier Industrie Et Sante
Ogilvy Renault Llp/s.e.n.c.r.l.,s.r.l.
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