Pge-1 containing lyophilized liposomes for use in the...

A - Human Necessities – 61 – K

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A61K 31/557 (2006.01) A61K 9/127 (2006.01)

Patent

CA 2240139

A method for the treatment of erectile dysfunction comprises instilling intra meatally an aqueous solution containing prostaglandin containing liposomes and a detergent for lysing the liposomes. A pharmaceutical composition for treating erectile dysfunction comprises a two component system. The first component comprises a predetermined amount of lyophilized prostaglandin containing liposomes. The second component comprises a predetermined volume of an aqueous solution containing a detergent for lysing the liposomes. Dissolution of the lyophilized prostaglandin containing liposomes yields a liquid composition suitable for application to the penis, to effect erection.

L'invention porte sur un traitement des troubles de l'érection consistant à injecter par le méat une solution aqueuse de liposomes contenant de la prostaglandine associée à un détergent de lyse des liposomes. Elle porte également sur une composition pharmaceutique de traitement desdits troubles consistant en un système à deux composants dont le premier est une quantité donnée de liposomes contenant de la prostaglandine lyophilisée et le second, une solution aqueuse de détergent de lyse des liposomes. La dissolution des liposomes contenant de la prostaglandine lyophilisée donne une composition liquide qui, appliquée au pénis, produit l'érection.

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