Pharmaceutical formulation comprising...

A - Human Necessities – 61 – K

Patent

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Details

IPC codes

A61K 31/505 (2006.01) A61K 31/27 (2006.01) A61K 31/519 (2006.01) A61K 45/06 (2006.01) A61P 25/22 (2006.01)

Type

Patent

Patent number

CA 2437085

Description

Pharmaceutical preparation comprising at least one phosphodiesterase V inhibitor have, and/or physiologically acceptable salts and/or solvates thereof and at least one endothelin receptor antagonist for the preparation of a medicament for the treatment of angina, high blood pressure, high pulmonary pressure, congestive heart failure (CHF), chronic obstructive pulmonary disease (COPD), cor pulmonale, dextrocardiac insufficiency, atherosclerosis, conditions of reduced patency of the heart vessels, peripheral vascular diseases, strokes, bronchitis, allergic asthma, chronic asthma, allergic rhinitis, glaucoma, irritable bowel syndrome, tumours, renal insufficiency, liver cirrhosis, erectile dysfunction and for the treatment of female sexual disorders.

L'invention concerne une préparation pharmaceutique comprenant au moins un inhibiteur de la phosphodiestérase V, et/ou des sels et/ou des solvates de celui-ci, acceptables au plan pharmaceutique, et au moins un antagoniste du récepteur de l'endothéline pour la préparation d'un médicament destiné au traitement de l'angine, de l'hypertension artérielle, de la pression pulmonaire élevée, de l'insuffisance cardiaque congestive (CHF), de la bronchopneumopathie chronique obstructive (COPD), du coeur pulmonaire, de la dextrocardie, de l'athérosclérose, de la liberté réduite des vaisseaux du coeur, des maladies vasculaires périphériques, de l'attaque, de la bronchite, de l'asthme allergique, de l'asthme chronique, de la rhinite allergique, du glaucome, du syndrome du côlon irritable, des tumeurs, de l'insuffisance rénale, de la cirrhose du foie, de la dysérection et pour le traitement des troubles sexuels chez la femme.

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