Pharmaceutically active compounds

Details Pharmaceutically active compounds Pharmaceutically active compounds

C - Chemistry, Metallurgy

07

K

C07K 5/06 (2006.01) A61K 31/352 (2006.01) A61K 31/7048 (2006.01) A61K 38/05 (2006.01) A61K 38/06 (2006.01) A61K 38/07 (2006.01) A61K 38/08 (2006.01) A61K 47/48 (2006.01) A61P 3/00 (2006.01) A61P 7/02 (2006.01) A61P 19/00 (2006.01) A61P 35/00 (2006.01) C07K 5/08 (2006.01) C07K 5/10 (2006.01) C07K 7/06 (2006.01)

Patent

CA 2675029

The invention relates to pharmaceutically active compounds comprising an isoflavone or isoflavone glycoside and an amino acid, peptide, or peptide derivative that is covalently bonded thereto, the peptide or peptide derivative containing 2 to 5 amino acids, as well as pharmaceutically acceptable salts or solvates of said compounds. Also disclosed are uses of such substances for producing pharmaceutical compositions, especially for the treatment of platelet aggregation and for tumor therapy. The invention can thus be used in the medical field and in the pharmaceutical industry. The compounds according to the invention are of general formula X-Pep, wherein X represents an isoflavone or isoflavone glycoside and Pep represents an amino acid or a peptide or peptide derivative containing 2 to 5 amino acids. X and Pep are covalently bonded or are linked by means of a linker system.

L'invention concerne des composés pharmaceutiquement actifs comprenant une isoflavone ou un glycoside d'isoflavone, et un aminoacide, un peptide ou un dérivé de peptide de 2 à 5 aminoacides lié par covalence avec le glycoside d'isoflavone, ainsi que des sels ou des solvates pharmaceutiquement acceptables de ces composés. L'invention concerne en outre des utilisations de tels produits pour la fabrication de compositions pharmaceutiques, en particulier pour le traitement de l'agrégation de thrombocytes et pour le traitement de tumeurs. Les domaines d'application de l'invention sont en conséquence la médecine et l'industrie pharmaceutique. Les composés selon l'invention répondent à la formule générale (I) X-Pep, dans laquelle X désigne une isoflavone ou un glycoside d'isoflavone, et Pep désigne un aminoacide ou un peptide ou un dérivé peptidique de 2 à 5 aminoacides, X et Pep étant liés par covalence ou par un système de linker.

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