C - Chemistry – Metallurgy – 07 – C
Patent
C - Chemistry, Metallurgy
07
C
C07C 217/60 (2006.01) A61K 31/192 (2006.01) A61K 31/22 (2006.01) A61P 1/12 (2006.01) A61P 3/04 (2006.01) A61P 3/10 (2006.01) A61P 13/10 (2006.01)
Patent
CA 2336853
The present invention provides novel phenoxyacetic acid derivatives represented by the above general formula and pharmaceutically acceptable salts thereof which have excellent .beta.3-adrenoceptor stimulating effects and are useful as agents for the prevention or treatment of obesity, hyperglycemia, the diseases caused by intestinal hypermotility, pollakiuria, urinary incontinence, depression, or the diseases caused by biliary calculi or hypermotility of biliary tract. (In the general formula, R1 represents a hydroxy group etc.; one of R2 and R3 is a hydrogen atom, a halogen atom etc., while the other is a hydrogen atom; R4 represents a halogen atom etc.)
On décrit de nouveaux dérivés d'acide phénoxyacétique de la formule générale (I) et des sels pharmacologiquement acceptables desdits dérivés, qui présentent un excellent effet de stimulation du récepteur beta 3-adrénergique et conviennent comme agents préventifs ou thérapeutiques contre l'obésité, l'hyperglycémie, les maladies causées par l'hypercinésie de l'intestin, la pollakiurie, l'incontinence urinaire, la dépression, la lithiase biliaire, ou les maladies causées par l'hypercinésie du tractus biliaire. Dans ladite formule, R<1> est hydroxyle ou analogue; l'un quelconque de R<2> et R<3> est hydrogène, halogéno ou analogue, l'autre étant hydrogène; et R<4> est halogéno ou analogue.
Akahane Masuo
Hirabayashi Akihito
Mukaiyama Harunobu
Muranaka Hideyuki
Sato Masaaki
Kirby Eades Gale Baker
Kissei Pharmaceutical Co. Ltd.
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