Pipecolic linker and its use for chemistry on solid support

Details Pipecolic linker and its use for chemistry on solid support Pipecolic linker and its use for chemistry on solid support

C - Chemistry, Metallurgy

07

D

C07D 211/60 (2006.01) C07B 61/00 (2006.01) C08F 8/10 (2006.01)

Patent

CA 2733967

The present invention relates to a pipecolic linker and its use as a solid- phase linker in organic synthesis. Said pipecolic solid-phase linker may be used for coupling functional groups chosen between primary amines, secondary amines, aro-matic amines, alcohols, phenols and thiols. In particular, said pipecolic solid-phase linker may be used for peptide or pseudopep-tide synthesis, such as the reverse N to C peptide synthesis or the retro-inverso peptide synthesis, or for the synthesis of small or-ganic molecules.

La présente invention concerne un lieur pipécolique et son utilisation en tant que lieur sur phase solide en synthèse organique. Ledit lieur pipécolique sur phase solide peut être utilisé pour le couplage de groupes fonctionnels choisis entre des amines primaires, des amines secondaires, des amines aromatiques, des alcools, des phénols et des thiols. En particulier, ledit lieur pipécolique sur phase solide peut être utilisé pour la synthèse de peptides ou de pseudo-peptides, telle que la synthèse de peptides inversés de N à C ou la synthèse de peptides rétro-inversés ou pour la synthèse de petites molécules organiques.

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