Piperazine derivatives for the treatment of hiv infections

Details Piperazine derivatives for the treatment of hiv infections Piperazine derivatives for the treatment of hiv infections

A - Human Necessities

61

K

A61K 31/496 (2006.01) A61K 31/18 (2006.01) A61K 31/495 (2006.01) C07D 213/64 (2006.01) C07D 215/20 (2006.01) C07D 215/26 (2006.01) C07D 217/02 (2006.01) C07D 231/12 (2006.01) C07D 231/56 (2006.01) C07D 235/08 (2006.01) C07D 239/74 (2006.01) C07D 249/08 (2006.01) C07D 263/56 (2006.01) C07D 295/192 (2006.01) C07D 401/12 (2006.01)

Patent

CA 2534866

This invention relates to a compound of formula (I) or pharmaceutically acceptable salts, solvates or derivatives thereof, wherein R1 to R5 are defined in the description, and to processes for the preparation thereof, intermediates used in their preparation, compositions containing them and the uses of such derivatives. The compounds of the present invention inhibit the interaction of gp 120 with CD4 and are therefore of use in the treatment of HIV, a retroviral infection genetically related to HIV, or AIDS.

La présente invention concerne un composé de formule (I) ou bien ses sels, solvates ou dérivés pharmaceutiquement acceptables, formule dans laquelle R?1¿ à R?5¿ sont tels que définis dans la description. L'invention concerne également des procédés pour leur préparation, des intermédiaires utilisés dans leur préparation, des compositions les contenant, ainsi que les utilisations de tels dérivés. Les composés décrits inhibent l'interaction de gp120 avec CD4 et sont donc utiles dans le traitement du VIH, des infections rétrovirales génétiquement apparentées au VIH, et du sida.

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