Piperidine derivatives

Details Piperidine derivatives Piperidine derivatives

C - Chemistry, Metallurgy

07

D

260/290.2, 260/2

C07D 211/58 (2006.01)

Patent

CA 1094059

ABSTRACT OF THE DISCLOSURE Piperidine derivatives, and process for their prepar- ation of formula: Image 1 wherein R represents a lower alkoxy or lower alkenyloxy group; R1 and R2, which may be the same or different, each represent a hydrogen or halogen atom, or a sulphamoyl, amino, lower alkyl- amino, di(lower)alkylamino, lower alkylsulphonyl or lower alkyl- sulphamoyl group, or a lower acylamino group in which the acyl moiety is derived from a carboxylic acid, the halogen atom or group represented by the symbol R1 being in the 3- or 4-position of the phenyl ring, with the proviso that R1 and R2 do not both represent hydrogen atoms; R3 represents a hydrogen atom or a lower alkyl group, and R4 represents a cycloalkyl group having from 3 to 7 carbon atoms in the ring optionally substituted by an alkyl group containing 1 to 3 carbon atoms, or R4 represents an adamantyl group; and pharmaceutically-acceptable acid add- ition salts and quaternary ammonium derivatives and N-oxides thereof. These compounds find use as agents to antagonize the effects of dopamine, and dopaminergic agents of endogenous or exogenous origin.

271918

Affiliated with

Also associated with

Rating

Piperidine derivatives does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Piperidine derivatives, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Piperidine derivatives will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-624694