C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 455/00 (2006.01) A61K 31/4375 (2006.01) A61K 31/55 (2006.01) A61P 3/06 (2006.01) A61P 3/10 (2006.01) A61P 9/02 (2006.01) A61P 15/10 (2006.01) A61P 25/00 (2006.01) A61P 25/14 (2006.01) A61P 25/16 (2006.01) A61P 25/18 (2006.01) A61P 25/22 (2006.01) A61P 25/24 (2006.01) A61P 25/28 (2006.01) C07D 455/03 (2006.01) C07D 471/04 (2006.01) C07D 471/14 (2006.01) C07D 491/14 (2006.01) C07D 491/147 (2006.01) C07D 495/14 (2006.01)
Patent
CA 2480695
The invention provides a compound of formula I, wherein X, Z, R1 to R10, R15, R16, m, n, r and t are as defined in claim 1, or a pharmaceutically acceptable salt or ester thereof, useful as an alpha-2 antagonist. The compounds of formula I can be used for the treatment of diseases or conditions where antagonists of alpha-2 adrenoceptors are indicated to be effective.
L'invention concerne un composé représenté par la formule (I), dans laquelle X, Z, R¿1? à R¿10?, R¿15?, R¿16?, m, n, r et t sont tels que définis dans la revendication 1, ou un ester ou un sel pharmaceutiquement acceptable de ce composé, lequel est utilisé comme antagoniste .alpha.2. Les composés représentés par la formule (I) peuvent être utilisés dans le traitement de maladies ou d'états pathologiques où les antagonistes des récepteurs .alpha.2-adrénergiques sont considérés efficaces.
Din Belle David
Haapalinna Antti
Jokela Reija
Karjalainen Arto
Ratilainen Jari
Orion Corporation
Robic
LandOfFree
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