Preparations for intraurethral administration

Details Preparations for intraurethral administration Preparations for intraurethral administration

A - Human Necessities

61

K

A61K 31/475 (2006.01) A61K 31/00 (2006.01) A61P 15/00 (2006.01) A61P 15/10 (2006.01) A61P 43/00 (2006.01) C07D 471/06 (2006.01)

Patent

CA 2353613

Medicinal compositions for intraurethral administration which contain, as the active ingredient, at least one member selected from among compounds having a cyclic GMP phosphodiesterase (hereinafter referred to simply as cGMP-PDE) inhibitory effect, in particular, pyridocarbazole derivatives represented by general formula (I), salts thereof and solvates thereof. These compositions potently and selectively inhibit cGMP-PDE without being affected by drug absorption caused by foods, exert little side effects, have a high safety, and exhibit excellent therapeutic effects on erectile dysfunction and female sexual dysfunction.

L'invention concerne des compositions médicinales destinées à être administrées par voie urétrale. Ces compositions contiennent, comme agent actif, au moins un élément choisi parmi des composés ayant un effet inhibiteur de la phosphodiestérase GMP cyclique (cGMP-PDE), notamment des dérivés de pyridocarbazole représentés par la formule générale (I), leurs sels et leurs solvates. Ces compositions présentent un effet inhibiteur puissant et sélectif sur cGMP-PDE sans être affectées par l'absorption de médicaments et de nourriture. Par ailleurs, ces compositions présentent peu d'effets secondaires, elles présentent une sécurité élevée et elles présentent de remarquables effets thérapeutiques sur la dysérection et la dysfonction sexuelle féminine.

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