Process for preparing 1,2-diacyl-sn-glycerols

C - Chemistry – Metallurgy – 07 – C

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

260/483.1, 260/4

C07C 69/30 (2006.01) C07C 69/58 (2006.01) C07F 5/02 (2006.01)

Patent

CA 1149818

ABSTRACT OF THE DISCLOSURE: The object of the present invention is a novel and simple process for the production of 1,2-diacyl-an-glycer- ols, wherein the acyl groups may be the same or different According to the invention D-mannitol is reacted with benzene boronic acid or a derivative thereof to form a D-mannitol- monobenzeneboronate which compound is acylated either to form, after removal of the benzeneboronate protective group, a 1,2,5,6-tetraacyl-D-mannitol with four identical acyl groups, or is acylated selectively in two stages, by first acylating the 1,6-hydroxy groups of the boronate protected D-mannitol to form, after removal of the boronate protection, a 1,6- diacyl-D-mannitol, which then is repeatedly reacted with a benzene boronic acid or a derivative thereof and then acylated in the 2- and 5- positions. After removal of the boronate protective group, the tetra-acylated D-mannitol obtained either in the one-stage or two-stage process is split by oxidation to form a 1,2-diacyl-glyceraldehyde which in turn is reduced to the corresponding 1,2-diacyl-sn-glycerol. By means of the invention it is thus possible to prepare 1,2-diacyl-sn- glycerols in which the acyl groups can be the same or dif- ferent.

374967

LandOfFree

Say what you really think

Search LandOfFree.com for Canadian inventors and patents. Rate them and share your experience with other people.

Rating

Process for preparing 1,2-diacyl-sn-glycerols does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Process for preparing 1,2-diacyl-sn-glycerols, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Process for preparing 1,2-diacyl-sn-glycerols will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFCA-PAI-O-950826

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.