Process for synthesizing a cetp inhibitor

Details Process for synthesizing a cetp inhibitor Process for synthesizing a cetp inhibitor

C - Chemistry, Metallurgy

07

D

C07D 263/22 (2006.01) A61K 31/421 (2006.01) A61P 9/10 (2006.01)

Patent

CA 2612142

An efficient process is disclosed for producing a compound that is an inhibitor of CETP. The last step of the process is the coupling of an oxazolidinone derivative with a biphenyl moiety to provide a compound of formula (I). In a specific embodiment of this synthesis, a crystalline product is produced which is characterized as a non-solvated crystalline polymorph.

L'invention concerne un procédé efficace permettant de produire un composé qui est un inhibiteur de CETP. La dernière étape du procédé est le couplage d'un dérivé d'oxazolidinone avec une fraction biphényle afin de fournir un composé représenté par la formule (I). Dans un mode de réalisation spécifique de cette synthèse, un produit cristallin caractérisé comme étant un polymorphe cristallin non solvaté est produit.

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