Process for the preparation of a piperazine derivative

Details Process for the preparation of a piperazine derivative Process for the preparation of a piperazine derivative

C - Chemistry, Metallurgy

07

D

C07D 413/06 (2006.01) C07D 241/04 (2006.01)

Patent

CA 2412873

(2R)-1-[3,5-Bis (trifluoromethyl) benzoyl]-4-[2-[(2S)-2-(methoxymethyl) morpholino]ethyl]-2-(3-hydroxy-4-methyl- benzyl) piperazine dihydrochloride can be prepared from (2R)-4-benzyl-1-[3,5-bis (trifluoromethyl) benzoyl]-2-(3- hydroxy-4-methylbenzyl) piperazine via debenzylation, N-alkylation, and conversion into hydrochloride.

On peut préparer (2R)-1-[3,5-bis(trifluorométhyle)benzoyle]-4-[2-[(2S)-2(méthoxyméthyle)morpholino]éthyle]-2-(3-hydroxy-4-méthyle-benzyle)piperazine dichlorhydrate à partir de (2R)-4-benzyle-1-[3,5-bis(trifluorométhyle)benzoyle]-2-(3-hydroxy-4-méthylbenzyle)piperazine par le biais de la débenzylation, la N-alkylation, et la conversion en chlorhydrate.

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