Processes for the synthesis of bazedoxifene acetate and...

Details Processes for the synthesis of bazedoxifene acetate and... Processes for the synthesis of bazedoxifene acetate and...

C - Chemistry, Metallurgy

07

D

C07D 209/12 (2006.01)

Patent

CA 2758109

Efficient processes for the synthesis of pharmaceutically useful compounds such as (1-[4-(2-azepan-1-yl-ethoxy)-benzyl] -2-(4-hydroxy-phenyl)-3-methyl-1H-indol-5-ol acetic acid commonly known as bazedoxifene acetate (Formula IX) using cyanomethoxybenzyl halides of Formula III, where X = Halogens e.g., Cl, F, Br, I; G = Any electron donating or electron withdrawing substituent.

L'invention porte sur des procédés efficaces pour la synthèse de composés pharmaceutiquement utiles tels que l'acide (1-[4-(2-azépan-1-yléthoxy)-benzyl]-2-(4-hydroxyphényl)-3-méthyl-1H-indol-5-olacétique, communément appelé acétate de bazédoxifène (Formule IX), à l'aide d'halogénure de cyanométhoxybenzyle de Formule III, où X = des halogènes, par exemple Cl, F, Br, I ; G = n'importe quel substituant donneur d'électrons ou attracteur d'électrons.

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