C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 417/04 (2006.01) A61K 31/428 (2006.01) A61P 35/00 (2006.01) C07D 413/04 (2006.01) C07D 417/14 (2006.01) C07D 513/04 (2006.01) C07D 521/00 (2006.01)
Patent
CA 2492964
A pharmaceutical composition comprising a pharmaceutically acceptable excipient and a compound of formula (I): wherein R1, R2 and R3 at each occurrence are independently selected from amino, aminosulfinyl, aminosulfonyl, aryl, azido, halogen, heteroalkyl, heteroaryl, hydrazinyl, hydrocarbyl, hydrogen, hydroxyl, nitro, nitroso, phosphate, phosphinate, phosphonate, phosphonium, phosphorothioate, phosphoryl, sulfamoyl, sulfate, sulfinic acid, sulfonamido, sulfonate, sulfonic acid, sulfonyl, sulfoxido, thiol, thioureido, and ureido, and R4 is selected from hydrogen, heteroalkyl, heteroaryl, and hydrocarbyl is described as useful in treatment of disorders associated with dysregulation of cell proliferation.
L'invention concerne des compositions pharmaceutiques de pyrazolybenzothiazole représentées par la formule (1). Ces compositions peuvent être constituées par des sels pharmaceutiquement acceptables. R?1¿, R?2¿ et R?3¿ sont dans chaque cas pris indépendamment parmi amino, aminosulfinyle, aminosulfonyle, aryle, azido, halogène, hétéroalkyle, hétéroaryle, hydrazinyle, hydrocarbyle, hydrogène, hydroxyle, nitro, nitroso, phosphate, phosphinate, phosphonate, phosphonium, phosphorothioate, phosphoryle, sulfamoyle, sulfate, acide sulfinique, sulfonamido, sulfonate, acide sulfonique, sulfonyle, sulfoxydo, thiol, thiouréido, et uréido, et R?4¿ et pris indépendamment parmi hydrogène, hétéroalkyle, hétéroaryle, et hydrocarbyle.
Chen Jianxin
Chopiuk Gregory B.
Daynard Timothy S.
Du Xinyao
Sviridov Serguei V.
Fetherstonhaugh & Co.
Qlt Inc.
Valocor Therapeutics Inc.
LandOfFree
Pyrazolylbenzothiazole derivatives and their use as... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Pyrazolylbenzothiazole derivatives and their use as..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Pyrazolylbenzothiazole derivatives and their use as... will most certainly appreciate the feedback.
Profile ID: LFCA-PAI-O-1531216