C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 471/04 (2006.01) A61K 31/4745 (2006.01) A61P 35/00 (2006.01)
Patent
CA 2673410
The present invention provides compounds of Formula I (wherein R, R1, R3, R4, X, and ring Y are as defined herein). The present invention also provides compositions comprising these compounds that are useful for treating cellular proliferative diseases or disorders associated with KSP kinesin activity and for inhibiting KSP kinesin activity.
La présente invention propose des composés de Formule I (dans laquelle R, R1, R3, R4, X et le noyau Y sont tels que définis présentement). La présente invention propose également des compositions comportant ces composés qui s'utilisent pour traiter les maladies de prolifération cellulaire ou des troubles associés à l'activité de la kinésine KSP et pour inhiber l'activité de la kinésine KSP.
Doll Ronald J.
Duca Jose S.
Lesburg Charles A.
Paliwal Sunil
Shih Neng-Yang
Ogilvy Renault Llp/s.e.n.c.r.l.,s.r.l.
Schering Corporation
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